Competitive routes to cyclizations of polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones with 3-aminopyrazoles into bioactive pyrazoloazines

Natalia A. Elkina; Yanina V. Burgart; Evgeny V. Shchegolkov; Olga P. Krasnykh; Vera V. Maslova; Galina A. Triandafilova; Sergey S. Solodnikov; Anna A. Muryleva; Maria A. Misiurina; Alexander V. Slita; Vladimir V. Zarubaev; Victor I. Saloutin

doi:10.1016/j.jfluchem.2020.109648

Competitive routes to cyclizations of polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones with 3-aminopyrazoles into bioactive pyrazoloazines

Natalia A. Elkina, Yanina V. Burgart, Evgeny V. Shchegolkov, Olga P. Krasnykh, Vera V. Maslova, Galina A. Triandafilova, Sergey S. Solodnikov, Anna A. Muryleva, Maria A. Misiurina, Alexander V. Slita, Vladimir V. Zarubaev, Victor I. Saloutin

Research output: Contribution to journal › Article › peer-review

3 Citations (Scopus)

Original language	English
Article number	109648
Number of pages	11
Journal	Journal of Fluorine Chemistry
Volume	240
DOIs	https://doi.org/10.1016/j.jfluchem.2020.109648
Publication status	Published - Dec 2020

Keywords

3-Aminopyrazoles
Analgesic and antiviral activities
Haloformic cleavage
N,N- and C,N-cyclization
Polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones
Pyrazolo[1,5-a]pyrimidines
Pyrazolo[3,4-b]pyridines
Toxicity
Pyrazolo[3,4-b] pyridines
DESIGN
ALPHA-AMINOAZOLES
DISCOVERY
PYRAZOLOPYRIDINE DERIVATIVES
POTENT
HETEROCYCLES
GROWTH
BIOLOGICAL EVALUATION
INHIBITORS
ANTAGONISTS

ASJC Scopus subject areas

Biochemistry
Inorganic Chemistry
Physical and Theoretical Chemistry
Environmental Chemistry
Organic Chemistry

WoS ResearchAreas Categories

Chemistry, Inorganic & Nuclear
Chemistry, Organic

Access to Document

10.1016/j.jfluchem.2020.109648

Cite this

Elkina, N. A., Burgart, Y. V., Shchegolkov, E. V., Krasnykh, O. P., Maslova, V. V., Triandafilova, G. A., Solodnikov, S. S., Muryleva, A. A., Misiurina, M. A., Slita, A. V., Zarubaev, V. V., & Saloutin, V. I. (2020). Competitive routes to cyclizations of polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones with 3-aminopyrazoles into bioactive pyrazoloazines. Journal of Fluorine Chemistry, 240, [109648]. https://doi.org/10.1016/j.jfluchem.2020.109648

Elkina, Natalia A. ; Burgart, Yanina V. ; Shchegolkov, Evgeny V. ; Krasnykh, Olga P. ; Maslova, Vera V. ; Triandafilova, Galina A. ; Solodnikov, Sergey S. ; Muryleva, Anna A. ; Misiurina, Maria A. ; Slita, Alexander V. ; Zarubaev, Vladimir V. ; Saloutin, Victor I. / Competitive routes to cyclizations of polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones with 3-aminopyrazoles into bioactive pyrazoloazines. In: Journal of Fluorine Chemistry. 2020 ; Vol. 240.

@article{dd82d2151b8549f5b1ea8631e2e95299,

title = "Competitive routes to cyclizations of polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones with 3-aminopyrazoles into bioactive pyrazoloazines",

keywords = "3-Aminopyrazoles, Analgesic and antiviral activities, Haloformic cleavage, N,N- and C,N-cyclization, Polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones, Pyrazolo[1,5-a]pyrimidines, Pyrazolo[3,4-b]pyridines, Toxicity, Pyrazolo[3,4-b] pyridines, DESIGN, ALPHA-AMINOAZOLES, DISCOVERY, PYRAZOLOPYRIDINE DERIVATIVES, POTENT, HETEROCYCLES, GROWTH, BIOLOGICAL EVALUATION, INHIBITORS, ANTAGONISTS",

author = "Elkina, {Natalia A.} and Burgart, {Yanina V.} and Shchegolkov, {Evgeny V.} and Krasnykh, {Olga P.} and Maslova, {Vera V.} and Triandafilova, {Galina A.} and Solodnikov, {Sergey S.} and Muryleva, {Anna A.} and Misiurina, {Maria A.} and Slita, {Alexander V.} and Zarubaev, {Vladimir V.} and Saloutin, {Victor I.}",

year = "2020",

month = dec,

doi = "10.1016/j.jfluchem.2020.109648",

language = "English",

volume = "240",

journal = "Journal of Fluorine Chemistry",

issn = "0022-1139",

publisher = "Elsevier BV",

}

Elkina, NA, Burgart, YV , Shchegolkov, EV, Krasnykh, OP, Maslova, VV, Triandafilova, GA, Solodnikov, SS, Muryleva, AA, Misiurina, MA, Slita, AV, Zarubaev, VV & Saloutin, VI 2020, 'Competitive routes to cyclizations of polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones with 3-aminopyrazoles into bioactive pyrazoloazines', Journal of Fluorine Chemistry, vol. 240, 109648. https://doi.org/10.1016/j.jfluchem.2020.109648

Competitive routes to cyclizations of polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones with 3-aminopyrazoles into bioactive pyrazoloazines. / Elkina, Natalia A.; Burgart, Yanina V.; Shchegolkov, Evgeny V.; Krasnykh, Olga P.; Maslova, Vera V.; Triandafilova, Galina A.; Solodnikov, Sergey S.; Muryleva, Anna A.; Misiurina, Maria A.; Slita, Alexander V.; Zarubaev, Vladimir V.; Saloutin, Victor I.

In: Journal of Fluorine Chemistry, Vol. 240, 109648, 12.2020.

Research output: Contribution to journal › Article › peer-review

TY - JOUR

T1 - Competitive routes to cyclizations of polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones with 3-aminopyrazoles into bioactive pyrazoloazines

AU - Elkina, Natalia A.

AU - Burgart, Yanina V.

AU - Shchegolkov, Evgeny V.

AU - Krasnykh, Olga P.

AU - Maslova, Vera V.

AU - Triandafilova, Galina A.

AU - Solodnikov, Sergey S.

AU - Muryleva, Anna A.

AU - Misiurina, Maria A.

AU - Slita, Alexander V.

AU - Zarubaev, Vladimir V.

AU - Saloutin, Victor I.

PY - 2020/12

Y1 - 2020/12

KW - 3-Aminopyrazoles

KW - Analgesic and antiviral activities

KW - Haloformic cleavage

KW - N,N- and C,N-cyclization

KW - Polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones

KW - Pyrazolo[1,5-a]pyrimidines

KW - Pyrazolo[3,4-b]pyridines

KW - Toxicity

KW - Pyrazolo[3,4-b] pyridines

KW - DESIGN

KW - ALPHA-AMINOAZOLES

KW - DISCOVERY

KW - PYRAZOLOPYRIDINE DERIVATIVES

KW - POTENT

KW - HETEROCYCLES

KW - GROWTH

KW - BIOLOGICAL EVALUATION

KW - INHIBITORS

KW - ANTAGONISTS

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UR - https://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcAuth=tsmetrics&SrcApp=tsm_test&DestApp=WOS_CPL&DestLinkType=FullRecord&KeyUT=000590770200001

U2 - 10.1016/j.jfluchem.2020.109648

DO - 10.1016/j.jfluchem.2020.109648

M3 - Article

AN - SCOPUS:85091777889

VL - 240

JO - Journal of Fluorine Chemistry

JF - Journal of Fluorine Chemistry

SN - 0022-1139

M1 - 109648

ER -

Competitive routes to cyclizations of polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones with 3-aminopyrazoles into bioactive pyrazoloazines

Keywords

ASJC Scopus subject areas

WoS ResearchAreas Categories

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Создание и развитие совместной лаборатории медицинской химии и перспективных органических материалов УрФУ – ИОС УрО РАН

Cite this

Competitive routes to cyclizations of polyfluoroalkyl-containing 2-tolylhydrazinylidene-1,3-diketones with 3-aminopyrazoles into bioactive pyrazoloazines

Keywords

ASJC Scopus subject areas

WoS ResearchAreas Categories

Access to Document

Other files and links

Fingerprint

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Создание и развитие совместной лаборатории медицинской химии и перспективных органических материалов УрФУ – ИОС УрО РАН

Cite this