Synthesis and biological evaluation of novel 5-aryl-4-(5-nitrofuran-2-yl)-pyrimidines as potential anti-bacterial agents

Egor V. Verbitskiy, Svetlana A. Baskakova, Natal'ya A. Gerasimova, Natal'Ya P. Evstigneeva, Natal'Ya V. Zil'Berberg, Nikolay V. Kungurov, Marionella A. Kravchenko, Marina G. Pervova, Gennady L. Rusinov, Oleg N. Chupakhin, Valery N. Charushin, S. N. Skornyakov

Research output: Contribution to journalArticleResearchpeer-review

9 Citations (Scopus)
Original languageEnglish
Pages (from-to)3003-3006
Number of pages4
JournalBioorganic and Medicinal Chemistry Letters
Volume27
Issue number13
DOIs
Publication statusPublished - 1 Jul 2017

Fingerprint

Nitrofurans
Spectinomycin
Pyrimidines
Neisseria gonorrhoeae
Staphylococcus aureus
Anti-Bacterial Agents
Pharmaceutical Preparations
In Vitro Techniques
pyrimidine
furan

Keywords

  • Antigonorrheal
  • Antimycobacterial
  • Nitrofuran
  • Nucleophilic aromatic substitution of hydrogen
  • Pyrimidine

ASJC Scopus subject areas

  • Biochemistry
  • Molecular Medicine
  • Molecular Biology
  • Pharmaceutical Science
  • Drug Discovery
  • Clinical Biochemistry
  • Organic Chemistry

WoS ResearchAreas Categories

  • Chemistry, Medicinal
  • Chemistry, Organic

Cite this

Verbitskiy, Egor V. ; Baskakova, Svetlana A. ; Gerasimova, Natal'ya A. ; Evstigneeva, Natal'Ya P. ; Zil'Berberg, Natal'Ya V. ; Kungurov, Nikolay V. ; Kravchenko, Marionella A. ; Pervova, Marina G. ; Rusinov, Gennady L. ; Chupakhin, Oleg N. ; Charushin, Valery N. ; Skornyakov, S. N. / Synthesis and biological evaluation of novel 5-aryl-4-(5-nitrofuran-2-yl)-pyrimidines as potential anti-bacterial agents. In: Bioorganic and Medicinal Chemistry Letters. 2017 ; Vol. 27, No. 13. pp. 3003-3006.
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keywords = "Antigonorrheal, Antimycobacterial, Nitrofuran, Nucleophilic aromatic substitution of hydrogen, Pyrimidine",
author = "Verbitskiy, {Egor V.} and Baskakova, {Svetlana A.} and Gerasimova, {Natal'ya A.} and Evstigneeva, {Natal'Ya P.} and Zil'Berberg, {Natal'Ya V.} and Kungurov, {Nikolay V.} and Kravchenko, {Marionella A.} and Pervova, {Marina G.} and Rusinov, {Gennady L.} and Chupakhin, {Oleg N.} and Charushin, {Valery N.} and Skornyakov, {S. N.}",
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Synthesis and biological evaluation of novel 5-aryl-4-(5-nitrofuran-2-yl)-pyrimidines as potential anti-bacterial agents. / Verbitskiy, Egor V.; Baskakova, Svetlana A.; Gerasimova, Natal'ya A.; Evstigneeva, Natal'Ya P.; Zil'Berberg, Natal'Ya V.; Kungurov, Nikolay V.; Kravchenko, Marionella A.; Pervova, Marina G.; Rusinov, Gennady L.; Chupakhin, Oleg N.; Charushin, Valery N.; Skornyakov, S. N.

In: Bioorganic and Medicinal Chemistry Letters, Vol. 27, No. 13, 01.07.2017, p. 3003-3006.

Research output: Contribution to journalArticleResearchpeer-review

TY - JOUR

T1 - Synthesis and biological evaluation of novel 5-aryl-4-(5-nitrofuran-2-yl)-pyrimidines as potential anti-bacterial agents

AU - Verbitskiy, Egor V.

AU - Baskakova, Svetlana A.

AU - Gerasimova, Natal'ya A.

AU - Evstigneeva, Natal'Ya P.

AU - Zil'Berberg, Natal'Ya V.

AU - Kungurov, Nikolay V.

AU - Kravchenko, Marionella A.

AU - Pervova, Marina G.

AU - Rusinov, Gennady L.

AU - Chupakhin, Oleg N.

AU - Charushin, Valery N.

AU - Skornyakov, S. N.

PY - 2017/7/1

Y1 - 2017/7/1

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KW - Antimycobacterial

KW - Nitrofuran

KW - Nucleophilic aromatic substitution of hydrogen

KW - Pyrimidine

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M3 - Article

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SP - 3003

EP - 3006

JO - Bioorganic and Medicinal Chemistry Letters

JF - Bioorganic and Medicinal Chemistry Letters

SN - 0960-894X

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